
(51) C 07 D 0407/14 (2006.01) Z C 07 D 0401/06 (2006.01)
(11) 01 162 201
(51) C 07 D 0409/04 (2006.01) Z A 61 K 0031/18 (2006.01)
(11) 01 029 541
(51) C 07 D 0409/06 (2006.01) Z C 07 D 0307/46 (2006.01)
(11) 00 962 456
(51) C 07 D 0409/12 (2006.01) Z C 07 D 0231/32 (2006.01)
(11) 01 481 970
(51) C 07 D 0409/14 (2006.01) Z C 07 D 0401/06 (2006.01)
(11) 01 322 635
(51) C 07 D 0409/14 (2006.01) Z C 07 D 0405/14 (2006.01)
(11) 01 330 453
(51) C 07 D 0413/04 (2006.01) Z A 61 K 0031/18 (2006.01)
(11)
01 029 541
(51) C07 D0413/06 (2006.01)
C07 D0401/06 (2006.01)
C07 D0403/06 (2006.01)
C07 D0471/04 (2006.01)
C07 D0413/14 (2006.01)
C07 D0495/04 (2006.01)
C07 F0007/18 (2006.01)
A61K0031/535 (2006.01)
A61K0031/495 (2006.01)
A61P0029/00 (2006.01)
A61P0003/00 (2006.01)
A61P0027/02 (2006.01)
C07 D0413/06 (2006.01)
C07 D0265/00 (2006.01)
C07 D0241/00 (2006.01)
(11) 01 140 924
(21) 99959751.1
(22)10.12.1999 (86)en
(43)10.10.2001(87)en
(24) 22.03.2006
(30)14.12.1998 AU PP770698
21.10.1999 AU PP356898
(54) PIPERAZIN-DERIVATE
(73)Astellas Pharma Inc.
3-11, Nihonbashi-Honcho 2-chome,
Chuo-ku, Tokyo (JP)
(72)TAKE, Kazuhiko
3-3-2-201, Kouyoudai
Tondabayashi-shi, Osaka 584-0082 (JP)
KONISHI, Nobukiyo
22-7, Aotanai
Nagaokakyo-shi, Kyoto 617-0811 (JP)
SHIGENAGA, Shinji
7-3-75-103, Yokoo
Suma-ku, Kobe-shi, Hyogo 654-0131 (JP)
KAYAKIRI, Natsuko
7-11, Aobaokaminami
Suita-shi, Osaka 565-0802 (JP)
AZAMI, Hidenori
3-5-2-1105, Sumiregaoka
Takarazuka-shi, Hyogo 665-0847 (JP)
EIKYU, Yoshiteru
559-1-303, Hourencho
Nara-shi, Nara 630-8113 (JP)
NAKAI, Kazuo
1-27-18-503, Mukonosohigashi
Amagasaki-shi, Hyogo 661-0032 (JP)
ISHIDA, Junya
4-20-608, Kumano-cho
Nishinomiya-shi, Hyogo 663-8103 (JP)
MORITA, Masataka
2-2-10-A103, Midorigaoka
Ikeda-shi, Osaka 563-0026 (JP)
(86)PCT/JP 1999/006943 (en)
(87)WO 2000/035915 22.6.2000
(51) C 07 D 0413/06 (2006.01) Z C 07 D 0413/06 (2006.01)
(11) 01 140 924
(51) C 07 D 0413/10 (2006.01) Z C 07 C 0271/16 (2006.01)
(11) 01 328 509
(51) C 07 D 0413/10 (2006.01) Z C 07 D 0405/10 (2006.01)
(11) 01 539 745
(51) C 07 D 0413/12 (2006.01) Z C 07 D 0231/32 (2006.01)
(11) 01 481 970
(51) C 07 D 0413/12 (2006.01) Z C 07 D 0403/12 (2006.01)
(11) 01 549 650
(21) 03807842.4
(22)06.10.2003 (86)de
(43)06.07.2005(87)de
(24) 22.03.2006
(30)08.10.2002 DE 10246890
(54) SUBSTITUIERTE
C-IMIDAZO[1,2-A]LPYRIDIN-3YL-METHYLAMINE
(73)Grünenthal GmbH
Zieglerstrasse 6
52078 Aachen (DE)
(72)SUNDERMANN, Bernd
Oppenhoffallee 83-85
52066 Aachen (DE)
HENNIES, Hagen-Heinrich
Eicherscheid 56
52152 Simmerath (DE)
SUNDERMANN, Corinna
Oppenhoffallee 83-85
52066 Aachen (DE)
OBERBÖRSCH, Stefan
Weidenweg 10
52074 Aachen (DE)
(86)PCT/EP 2003/011011 (de)
(87)WO 2004/033453 22.4.2004
(51) C 07 D 0471/04 (2006.01) Z C 07 D 0471/04 (2006.01)
(11) 01 549 650
(51) C 07 D 0471/04 (2006.01) Z C 07 D 0413/06 (2006.01)
(11) 01 140 924
(51) C07 D0471/04 (2006.01)
A61K0031/437 (2006.01)
A61P0025/00 (2006.01)
C07 D0471/04 (2006.01)
C07 D0235/00 (2006.01)
C07 D0221/00 (2006.01)
(11) 01 200 433
(21) 00948852.9
(22)20.07.2000 (86)en
(43)02.05.2002 (87)en
(24) 22.03.2006
(30)02.08.1999 US 146731
(54) C-6 RINGSUBSTITUIERTE
PYRIDO[1,2-A]BENZIMIDAZOLDERIVATE ZUR
BEHANDLUNG VON STÖRUNGEN DES ZENTRALEN
NERVENSYSTEMS
(73)Ortho-McNeil Pharmaceutical, Inc.
920 U.S. Route No.202
Raritan, NJ 08869 (US)
(72)REITZ, Allen, B.
109 Greenbrier Road
Lansdale, PA 19446 (US)
NORTEY, Samuel, O.
7423 Euston Road
Elkins, PA 19027 (US)
SANFILIPPO, Pauline
7 Quimby Lane
Flemington, NJ 08822 (US)
SCOTT, Malcolm, K.
1036 Beverly Way
Lansdale, PA 19446 (US)
(86)PCT/US 2000/019882 (en)
(87)WO 2001/009132 8.2.2001
(51) C 07 D 0471/04 (2006.01) Z C 07 D 0471/04 (2006.01)
(11) 01 200 433
(51) C07 D0471/04 (2006.01)
A61K0031/5025 (2006.01)
(11) 01 244 660
(21) 00987932.1
(22)19.12.2000 (86)en
(43)02.10.2002 (87)en
(24) 22.03.2006
(30)23.12.1999 US 171906 P
29.09.2000 US 236881 P
(54) METHODEN UND ZUSAMMENSETZUNGEN ZUR
BEHANDLUNG VON SCHMERZEN
(73)AstraZeneca AB
151 85 Södertälje (SE)
(72)URBANEK, Rebecca Ann AstraZeneca
1800 Concord Pike, P.O. Box 15437
Wilmington, DE 19850-5437 (US)
BARE, Thomas, Michael
1057 Windy Knoll Road
(11) 00 979 823
(51) C 07 D 0413/12 (2006.01) Z C 07 D 0403/12 (2006.01)
(11) 00 979 823
(51) C 07 D 0413/14 (2006.01) Z C 07 D 0405/14 (2006.01)
(11) 01 330 453
(51) C 07 D 0413/14 (2006.01) Z C 07 D 0413/06 (2006.01)
(11) 01 140 924
(51) C 07 D 0413/14 (2006.01) Z C 07 D 0401/06 (2006.01)
(11) 01 162 201
(51) C 07 D 0417/06 (2006.01) Z C 07 K 0005/078 (2006.01)
(11) 00 933 379
(51) C 07 D 0417/06 (2006.01) Z C 07 D 0417/08 (2006.01)
(11) 01 272 488
(51) C07 D0417/08 (2006.01)
A61P0037/00 (2006.01)
C07 D0417/06 (2006.01)
C07 D0417/14 (2006.01)
A61K0031/427 (2006.01)
(11) 01 272 488
(21) 01914905.3
(22)19.03.2001(86)en
(43)08.01.2003 (87)en
(24) 22.03.2006
(30)23.03.2000 US 191668 P
(54) TRIARYLSUBSTITUIERTE ETHANE ALS PDE4
INHIBITOREN
(73)Merck Frosst Canada & Co.
16711 Trans-Canada Highway
Kirkland, Quebec H9H 3L1 (CA)
(72)FRIESEN, Richard
16711 Trans-Canada Highway
Kirkland, Québec H9H 3L1 (CA)
DUCHARME, Yves
16711 Trans-Canada Highway
Kirkland, Québec H9H 3L1 (CA)
COTE, Bernard
16711 Trans-Canada Highway
Kirkland, Québec H9H 3L1 (CA)
BLOUIN, Marc
16711 Trans-Canada Highway
Kirkland, Québec H9H 3L1 (CA)
MARTINS, Evelyn
16711 Trans-Canada Highway
Kirkland, Québec H9H 3L1 (CA)
GUAY, Daniel
16711 Trans-Canada Highway
Kirkland, Québec H9H 3L1 (CA)
HAMEL, Pierre
16711 Trans-Canada Highway
Kirkland, Québec H9H 3L1 (CA)
GIRARD, Mario
16711 Trans-Canada Highway
Kirkland, Québec H9H 3L1 (CA)
FRENETTE, Richard
16711 Trans-Canada Highway
Kirkland, Québec H9H 3L1 (CA)
LALIBERTE, Sebastien
16711 Trans-Canada Highway
Kirkland, Québec H9H 3L1 (CA)
(86)PCT/CA 2001/000365 (en)
(87)WO 2001/070738 27.9.2001
(51) C 07 D 0417/12 (2006.01) Z C 07 D 0231/32 (2006.01)
(11) 01 481 970
(51) C 07 D 0417/12 (2006.01) Z C 07 D 0403/12 (2006.01)
(11)
00 979 823
(51) C 07 D 0417/12 (2006.01) Z C 07 D 0403/12 (2006.01)
(11) 00 979 823
(51) C 07 D 0417/14 (2006.01) Z C 07 D 0401/06 (2006.01)
(11)
01 322 635
(51) C 07 D 0417/14 (2006.01) Z C 07 D 0417/08 (2006.01)
(11) 01 272 488
(51) C07 D0471/04 (2006.01)
A61K0031/437 (2006.01)
A61P0025/00 (2006.01)
A61P0035/00 (2006.01)
C07 D0471/04 (2006.01)
C07 D0235/00 (2006.01)
C07 D0221/00 (2006.01)
935
31.3.2006 +pat+6
Komentáře k této Příručce